Drugs Affecting the CNS
CLASS |
DRUG |
General Anesthetics |
Halothane, Isoflurane, Nitrous Oxide, Ketamine |
Local Anesthetics |
Benzocaine |
Neuromuscular Blockers |
Succinylcoline |
Procedural Sedation |
Benzodiazepine (Midazolam), Opioids (morphine/fentanyl), Propofol + fentanyl or midazolam |
Analgesic Opioids
CLASS |
DRUG |
Agonists |
Codeine, Hydrocodone, Morphine, Hydromorphone, Oxycodone, Meperidine, Fentanyl & Methadone |
Ceiling Effect |
Codiene Phosphate, Pentazocine, Nalbuphine |
Agonist-Antagonist |
Pentazocine, Butorphanol, Nalbuphine, Buprenorphine |
Antagonist |
Naloxone, Naltrexone |
Antiparkinsonian Drugs
CLASS |
DRUG |
Anti-Cholinergic |
Benzotropine, Diphenhydramine (anti-histamine) |
Catechol-o-methyl Transferase |
Entacapone |
Dopamine Agonist (DA) |
Bromocriptine, Pramipexole, Ropinirole, Rotigotine |
Levodopa (dopamine precursor) |
Levodopa |
MAO-B Inhibitors |
Rasagiline, Selegiline |
NMDA Antagonist |
Amantadine |
Antitubercular Drugs
CLASS |
DRUG |
Isoniazid |
Isoniazid (INH) |
Vitamin B6 |
Pyridoxine |
Rifampin |
Rifampin (RMP) |
Pyrazinamide |
Pyrazinamide (PZA) |
Ethambutol |
Ethambutol (EMB) |
Antifungal Drugs
CLASS |
DRUG |
Systemic Fungal Disease |
Amphotericin B |
Azole |
Clotrimazole |
Systemic and Superficial Fungal |
Fluconazole, Nystatin |
Antiprotozoans
CLASS |
DRUG |
Antimalarial |
Chloroquine, Hydrochloroquine, Mefloquine, Atovaquonel, Proquanil |
Trichomoniasis |
Metronidazole |
Beaver Fever Giardiasis |
Metronidazole or Paromomycin |
Immunosuppressants and Immunizations
CLASS |
DRUG |
Calcineurin Inhibitors |
Cyclosporine (with azathioprine) |
Biologics |
Derived from living cells |
Monoclonal Antibodies |
Adalimumab |
Hepatitis B |
Recombivax HB, Engerix-B |
Herpes |
Shingrix |
Anti-Cancer |
Gradasil 9 |
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CNS Depressants
CLASS |
DRUG |
Benzodiazepines |
Lorazepam, Clonazepam, Diazepam, Flunitrazepam, Midazolam, Alprazolam |
Non-Benzodiazepines |
Zopiclone, Buspirone Hydrocholride, Zolipidam |
Barbituates |
Phenobarbital, Secobarbital, Thiopental |
Muscle Relaxants |
Baclofen, Cyclobenzaprine, Dantrolene |
Serotonin Agonists |
Sumatriptan, Almotriptan, Eletriptan, Naratriptan, Rizatriptan, Zolmitriptan |
Non-Opioid Analgesics
CLASS |
DRUG |
NSAIDS |
Acetaminophen, ASA (Asprine), Ibuprofen, Naproxen, COX-2 Inhibitors, Tramadol Hydrochloride |
Antiepileptic Drugs
CLASS |
DRUG |
Antiepileptics |
Phenytoin, Carbazaepine, Phenobarbital, Gabapentin |
ANS Drugs
CLASS |
DRUG |
Adrenergics |
Salbbutamol, Vasopressors, Adrenergic Decongestants |
Non-Adrenergics |
Alpha and Beta cells |
Cholinergics |
Bathanechal, Acetylcholinesterase Inhibitor, Nicotine |
Non-Cholinergics |
Atropine, Benzotropine, Oxybutynin, Ipratropium Bromide |
Antiviral Drugs
CLASS |
DRUG |
CMV |
Glanciclovir, Valganciclovir |
Non HIV (Herpes Virus) |
Acyclovir, Valacyclovir |
Non HIV (Influenza) |
Oseltamivir Phosphate, Zanamivir |
Non HIV (COVID-19) |
Remdesvir, PAXLOVID (Nirmatrelvir & Ritonavir) |
Pre-Exposure (HIV) Prophylaxis (PrEP) |
Truvada & Descovy |
Antiretrovirals HIV |
Abacavir, Emtricitabine, Tenoforvir, Efavirenz, Etravirine, Nevirapine, Atazanavir, Durunavir, Ritonavir, Enfuvirtide, Maraviroc, Raltegravir |
Post-Exposure Prophaylaxis (PEP) |
Tenofovor, Emtricitabine, Raltgravir, Dolutegravir |
Antihelmintics
CLASS |
DRUG |
Anthelmintics |
Mabendazole, Praziquantel, Pyrantel Pamoate |
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